Presynaptic Receptors and Neuronal Transporters. Official Satellite Symposium to the IUPHAR 1990 Congress Held in Rouen, France, on 26–29 June 1990

Content: 
ADVANCES IN THE BIOSCIENCES, Page ii
Front Matter, Page iii
Copyright, Page iv
Preface, Pages xix-xx, S.Z. Langer, A.M. Galzin, J. Costentin
Physiological and Pharmacological Relevance of Presynaptic Receptors in Neurotransmission, Pages 1-5, S.Z. Langer, I. Angel, H. Schoemaker
Pre- and Postjunctional Muscarinic Receptors in the Guinea-pig Trachea, Pages 7-10, H. Kilbinger, D. Wolf, G. D'Agostino
Presynaptic α-autoadrenoceptors on Peripheral Noradrenergic Neurones of Newborn Rabbits and Dogs, Pages 11-14, S. Guimarães, M.Q. Paiva, D. Moura, M.J. Vaz-da-Silva
Cholinergic—Adrenergic Presynaptic Interactions in the Heart and Characterization of the Receptors Involved, Pages 15-18, E. Muscholl, A. Habermeier-Muth, U. Altes, K. Forsyth
Structural Requirements for DA2 (peripheral) Dopamine Receptor Agonist Activity, Pages 19-22, J.D. Kohli, P.T. Horn
α2-adrenoceptor Modulation of Noradrenaline Release in Human and Rabbit Renal Arteries: Clonidine Acts as a Partial Agonist, Pages 23-24, L.C. Rump, G. Ruff, P. Schollmeyer
Effect of α2-adrenoceptor Antagonists on Norepinephrine Release and Inhibition of Insulin Secretion During Pancreatic Nerve Stimulation. Interactions at Pre- and Postsynaptic Sites, Pages 25-26, N. Duval, I. Angel, A. Oblin, M.T. Eon, S.Z. Langer
Antagonist Activity of SL 84.0418 and Idazoxan at Pre and Postsynaptic α2-adrenoceptors, Pages 27-28, H. Schoemaker, A. Grosset, I. Angel, S.Z. Langer
Does the Distance Between Nerve Varicosities and Adrenoceptors Play Any Role in the Relative Contribution of ATP/Noradrenaline for Postjunctional Response?, Pages 29-30, J. Gonçalves, F. Carvalho, S. Guimarães
In vivo Presynaptic Interaction Between 5-HT and Adrenergic Antagonists on Noradrenergic Neurotransmission, Pages 31-32, M. Davy, F. Beslot, M. Midol-Monnet, M. Heimburger, Y. Cohen
Activity of N-ethyl-norarecaidine Propargyl Ester and (R)-nipecotic Acid Ethyl Ester at Pre- and Postsynaptic Muscarinic Receptor Subtypes, Pages 33-34, M. Eltze, F. Dörje, H. Tietz, A. Immel, E. Mutschler, G. Lambrecht
Effects of Neuromuscular Blocking Agents on Neuronal Nicotine Receptors of Motor Nerves: Blockade of Nicotinic Autofacilitation and Backfiring, Pages 35-36, I. Wessler, E. Jung, K. Wagenmann, T. Vogt, R. Besser
A Rapid in vitro Assay of the Histamine H3-receptor: Inhibition of Electrically Evoked Contractions of Guinea-pig Ileum Preparations, Pages 37-38, G.J. Menkveld, H. Timmerman
Factors Influencing the Function of Presynaptic α2-adrenoceptors in Rat Brain, Pages 39-42, P.J. Hollingsworth, C.B. Smith
Presynaptic Dopaminergic Autoreceptors as Targets for Drugs, Pages 43-46, A. Carlsson
DOPA Itself Facilitates Noradrenaline Release via Presynaptic β-adrenoceptors in Rat Hypothalamic Slices — DOPA is Probably a Neuroactive Substance, Pages 47-50, Y. Misu, Y. Goshima, S. Nakamura
The Third Dopamine Receptor (D3) as an Autoreceptor, Pages 51-54, J.C. Schwartz, P. Sokoloff, B. Giros, M.P. Martres, M.L. Bouthenet
Terminal Dopaminergic Autoreceptors are of Minor Importance for the Sedation Produced by DA Receptor Agonists in Rats, Pages 55-58, S. Ahlenius, V. Hillegaart, L. Svensson
Modulation of 5-HT Release by Presynaptic Inhibitory and Facilitatory 5-HT Receptors in Brain Slices, Pages 59-62, A.M. Galzin, S.Z. Langer
Modulation of 5-hydroxytryptamine and Noradrenaline Release in the Brain and Retina via Presynaptic Heteroreceptors: Some New Aspects, Pages 63-66, M. Göthert, E. Schlicker, K. Fink, G. Molderings
Autoreceptors and Heteroreceptors Evidenced by Histamine H3 Receptor Ligands, Pages 67-70, M. Garbarg, J.M. Arrang, C. Llorens-Cortes, H. Pollard, A. Rouleau, J.C. Schwartz, M.D. Trung Tuong, R. Lipp, H. Stark, W. Schunack, J.M. Lecomte
Somato-dendritic 5-HT1A Autoreceptors in the Dorsal Raphe Nucleus; Pharmacological and Functional Properties, Pages 71-74, M. Hamon, S. El Mestikawy, L. Lanfumey, J. Adrien, C.M. Fattaccini, H. Gozlan
Autoreceptor-mediated Control of Serotonin Release in the Rat Brain in vivo, Pages 75-78, B. Scatton, L. Rouquier, G. Bonvento, A. Serrano, P. Blier
Effects of α2-adrenoceptor Agonist and Antagonist on Spatial Memory in Rats, Pages 79-80, M.M. Airaksinen, S.A. Nieminen, E.J. MacDonald, J. Sirviö, P.J. Riekkinen Jr.
Modulation of the Ca2+-evoked Release of Dopamine from Synaptosomes, Pages 81-83, N. Weiner, J.F. Bowyer, J. Masserano
Evidence Against a Direct Link Between Serotonin Uptake Sites and Presynaptic Serotonin Autoreceptors, Pages 85-86, N. Limberger, E. Singer, K. Starke
A Comparison of Presynaptic Serotonin Autoreceptors in Rabbit, Rat and Guinea-pig Brain Cortex, Pages 87-88, R. Deicher, N. Limberger, K. Starke
Serotonergic Modulation of the Release of [3H]GABA from Guinea-pig Hippocampal Synaptosomes, Pages 89-90, I. Cloez, C. Harel-Dupas, G. Fillion
Pre- and Postsynaptic Location of 5-HT3 Receptors in the Rat Spinal Cord, Pages 91-92, A.M. Laporte, M.C. Lombard, S. Bourgoin, D. Verge, H. Gozlan, M. Hamon
Distribution of [3H]SCH 23390 Binding Sites in the Human Substantia Nigra, Pages 93-94, F. Thibaut, E.C. Hirsch, R. Raisman, F. Javoy-Agid, Y. Agid
Presynaptic Regulation of Dopamine Release from Synaptosomes of the Rat Striatum is Controlled by Different Types of Glutamate Receptors, Pages 95-96, J.M. Desce, G. Godeheu, A. Chéramy, J. Glowinski
Microdialysis Studies of the Effects of Local Apomorphine Infusions on Dopamine Release in Rat Striatum, Pages 97-98, M. Goiny, T. Guix, M. Herrera-Marschitz, U. Ungerstedt
Dopaminergic Hetero-regulation of Striatal μ-Opiate Receptors: Further Evidence for Their Postsynaptic Location, Pages 99-100, F. Trovero, D. Herve, M. Desban, J. Glowinski, J.P. Tassin
Presynaptic Modulation of Striatal Dopamine Release by Enkephalins, Pages 101-102, N. Dourmap, A. Michael-Titus, J. Costentin
Modulation of Dopamine and Acetylcholine Release in the Rabbit Caudate Nucleus by Opioids: Receptor Type and Interaction with Autoreceptors, Pages 103-104, R. Jackisch, H. Hotz, G. Hertting
Presynaptic Autoreceptors May Control the Release of Metenkephalin from the Rat Spinal Cord, Pages 105-106, E. Collin, S. Bourgoin, D. Chantrel, J.J. Benoliel, A. Mauborgne, M. Hamon, F. Cesselin
Involvement of NMDA Receptors in the Presynaptic Regulation of Dopamine Release in Striosome-and Matrix-enriched Areas of the Rat Striatum, Pages 107-108, Marie-Odile Krebs, Marie-Lou Kemel, Marcel Desban, Jacques Glowinski, Christian Gauchy
Inhibition of Synaptosomal Tyrosine Hydroxylase by Dopamine Autoreceptors: Role of Ca2+ and K+, Pages 109-110, Pierluigi Onali, Enrica Mosca, Maria C. Olianas
Dopaminergic Modulation of Striatal Sensory Responses, Pages 111-112, T.I. Lidsky, C. Manetto, S.P. Banerjee
Selective Presynaptic Dopamine Agonist Treatment of Schizophrenia with BHT-920, Pages 113-116, Peter Winckler, Mathias Bartels
Effects of the Antiparkinsonian Drugs Amantadine and Memantine on Striatal Neurotransmitter Release in vitro, Pages 117-118, A. Lupp, T. Link, G. Hertting, R. Jackisch, T.J. Feuerstein
Transmitter Interactions in Striatum May Occur via Effects on High Affinity Transporters, Pages 119-120, G. Lonart, S. Bernath, M.J. Zigmond
A Comparison of the Effect of Baclofen on Radiolabelled GABA and Noradrenaline Release in Rat Cortical Slices, Pages 121-122, Christine Ennis, Michael C.W. Minchin
Effects of Chronic Treatment with Flunitrazepam on GABAA, Adenosine and Glutamate Receptor Plasticity in Rats, Pages 123-124, M. Baraldi, P. Zanoli, A. Giacobazzi, G. Vaccari, R. Avallone
Modulation of N-Methyl-D-Aspartate (NMDA)-stimulated Noradrenaline Release in Rat Brain Cortex by Presynaptic α2-adrenoceptors and Histamine H3 Receptors, Pages 125-126, K. Fink, E. Schlicker, M. Göthert
Noradrenaline Release in the Pig Retina and Its Histamine H3 Receptor-mediated Inhibition, Pages 127-128, E. Schlicker, M. Göthert
Structure and Function of the GABA Reuptake System, Pages 129-134, Baruch I. Kanner
Energizing the Vacuolar System of Eukaryotic Cells, Pages 135-138, Nathan Nelson
The Molecular Size of the Neuronal Noradrenaline Carrier, Pages 139-142, H. Bönisch, J. Michael-Hepp, B. Blum, G. Martiny-Baron
Identification and Regulation of High-affinity-choline Transporter, Pages 143-146, M. Knipper
Ketanserin as a Ligand of the Vesicular Monoamine Transporter, Pages 147-150, J.P. Henry, B. Gasnier, M.F. Isambert, F. Darchen, D. Scherman
Dopamine Transporter — Cocaine Receptor: Characterization and Purification, Pages 151-154, R. Simantov, R. Vaughan, R. Lew, A. Wilson, M.J. Kuhar
Characterization and Purification of the Serotonin Transporter Located at the Cytoplasmic Membrane of Human Platelets: A Three-step Strategy, Pages 155-158, J.M. Launay, C. Chopin-Robert, C. Geoffroy, D. Bondoux, D. Lamblin, M.L. Giron, V. Mutel, M.H. Buc-Caron, L. Lasneret, O. Kellermann, M. Da Prada, J.E. Alouf
Molecular Characterization of the Neuronal Sodium-ion Coupled 5-hydroxytryptamine Transporter, Pages 159-162, D. Graham, H. Esnaud, S.Z. Langer
Kinetic Analyses of the Na+ and Cl–-Dependences of the Synaptosomal Specific Uptake of 3H Dopamine, Pages 163-164, N. Chab, J.-J. Bonnet, J. Costentin
Localization of Dopamine Uptake Complex by BTCP on Rat Brain Sections and Dopaminergic Neurons in vitro, Pages 165-166, C. Cerruti, J.-M. Kamenka, A. Privat
In vivo Binding of [3H]GBR 12783 in Mouse Brain — Characteristics of the Labelling of Striatal Dopamine Uptake Sites, Pages 167-168, J.-M. Vaugeois, J.-J. Bonnet, J. Costentin
[3H]GBR12935 Binds to Membrane from the Human Platelet, Pages 169-170, Brian Dean, David L. Copolov
Dopamine Transporter in Aging, Pages 171-173, Ikuya Shimizu, Chandan Prasad
Sodium Dependent, High Affinity Choline Transport Expressed in Oocytes, Pages 175-176, S. O'Regan, S. Birman, F.M. Meunier
Comparison of the Effects of Vesamicol and of Cetiedil Analogues on Acetylcholine Release and Vesicular Acetylcholine Transport, Pages 177-178, M.F. Diebler, Y. Morot Gaudry-Talarmain, J.C. Lancelot, M. Robba, J.L. Morgat, M. Israel
Dopamine Modulates [3H]BTCP (a Phencyclidine Derivative) Binding to the Dopamine Uptake Complex, Pages 179-180, J. Vignon, T. Maurice, G. Barbanel, J.M. Kamenka
The Heterogeneous Labelling with 3H-noradrenaline of the Incubated Vas Deferens of the Rat, Pages 181-184, U. Trendelenburg, C.-L. Schönfeld, T. Halbrügge, E. Schömig
Alterations in Platelet [3H]-Imipramine Binding, 5HT Uptake and Plasma α1-acid Glycoprotein Concentrations in Patients with Major Depression, Pages 185-188, David L. Knight, Theodore A. Slotkin, Lawrence R. Meyerson, K. Ranga, R. Krishnan, Charles B. Nemeroff
Ionic and Temperature Dependences of the 3H Dopamine Specific Uptake and 3H GBR 12783 or 3H Mazindol Specific Binding on the Dopamine Neuronal Carrier, Pages 189-192, J.-J. Bonnet, S. Benmansour, N. Chab, J. Costentin, E.M. Parker, L.X. Cubeddu
Dynamic Properties of Monoamine Storage Vesicles: Pharmacological and Physiological Implications, Pages 193-196, C. Desnos, F. Darchen, Y. Masuo, W. Rostene, D. Scherman
GABA Uptake Inhibitors: Kinetics and Molecular Pharmacology, Pages 197-200, O.M. Larsson, E. Falch, A. Schousboe, P. Krogsgaard-Larsen
Coexistence of More Than One Neurotransmitter Uptake System on the Same Nerve Terminal in the Brain, Pages 201-205, M. Raiteri, G. Bonanno, M. Pende, S. Setti
Peptidergic Regulation of Striatal Dopamine Transporter Complex, Pages 207-211, Chandan Prasad
Different Interactions of Citalopram with the Prejunctional Effects of Serotonin in Peripheral Tissues, Pages 213-217, E. Adler-Graschinsky, N.V. Butta, A.B. Elgoyhen, P.S. Lorenzo
Evolution of the Vesicular Monoamine Transporter During Ageing in the Rat Brain: a Quantitative Autoradiographic Study with 3H Dihydrotetrabenazine, Pages 219-220, I. Leroux-Nicollet, J. Costentin
Influence of the Oxygen Disponibility on the Efficiency of the Neuronal Dopamine Uptake Complex, Pages 221-222, B. Naudin, Ch. Saligaut, J. Costentin
Differences in Behavioural Responses Elicited by Dexamphetamine and the Pure Dopamine Uptake Inhibitor GBR 12783, Pages 223-224, D. Duterte-Boucher, J. Costentin
Protection of the Synaptosomal 5-HT Uptake System by a Ginkgo Biloba Extract (GBE 761), Pages 225-226, C. Ramassamy, J. Costentin
The Binding of Noradrenaline to the Substrate Recognition Site of the Neuronal Noradrenaline Carrier (Uptake1) Depends on Sodium and Chloride, Pages 227-228, E. Schömig
In vivo Distribution of Radiolabelled Citalopram in Brain as a Marker of 5-HT Uptake Sites for PET, Pages 229-230, S.P. Hume, J.E. Cremer, V.W. Pike, C. Pascali, A.A. Lammertsma, R. Dolan, C.J. Bench
Relationship of [3H]Paroxetine Binding and 5-HT Recognition Sites on the Neuronal Serotonin Transporter, Pages 231-232, B. Foy, A. Hepner, P.D. Hrdina
Effects of Repeated Administration of Antidepressants on Serotonin Uptake Sites Measured Using [3H]Cyanoimipramine Autoradiography, Pages 233-234, D.J. Brunswick, G.B. Kovachich, C.E. Aronson, A. Frazer
Rapid Changes in 3H-Imipramine Binding in Platelets of Depressed Patients After Amineptine Treatment, Pages 235-236, R. Jeanningros, B. Gronier, J.M. Azorin, R. Tissot
Brain 5-HT Uptake Sites, Labelled with [3H]Paroxetine, in Depressed Suicides, Pages 237-238, K.M. Lawrence, F. De Paermentier, S.C. Cheetham, M.R. Crompton, C.L.E. Katona, R.W. Horton
Pinoline, the Natural Ligand of Serotonin Transporter in Retina and Pineal Gland, Pages 239-240, M.M. Airaksinen, E. Kari
Differential Interaction of Phencyclidine (PCP) with the Dopamine Uptake Complex and the PCP Receptor in vivo, Pages 241-242, T. Maurice, J. Vignon, J.-M. Kamenka, J.-L. Pirat, R. Chicheportiche
The Uptake of the Amino Acid L-alanine on Its Inhibitory Presynaptic Effects in Rat Isolated Atria, Pages 243-244, N.V. Butta, D.S. Hansen, E. Adler-Graschinsky
Role of Omega (BZD) Sites of the GABAA Receptor Macromolecular Complex in the Modulation of Serotonin Release, Pages 245-248, A. Lista, S. Arbilla, S.Z. Langer
Mechanisms of Inhibition of Transmitter Release by Adenosine Analogs, Pages 249-252, B.B. Fredholm, P.-S. Hu, I. van der Ploeg, M. Dunér-Engström, T.V. Dunwiddie
Dependence of the A1-adenosine Receptor-mediated Inhibition of [3H]Noradrenaline Release in Hippocampus on the Stimulation Conditions, Pages 253-256, C. Allgaier, R. Greber, M. Hippach, G. Hertting
Modulation of [3H]-serotonin Release in Rat Spinal Cord Synaptosomes via Dihydropyridine-sensitive Calcium Channels and Protein Kinase C, Pages 257-260, D.J. Jones, V.C. Gandhi
G-proteins and Prejunctional α-adrenoceptors, Pages 261-264, T.V. Murphy, H. Majewski
Opioid Inhibition of Oxytocin Release, but not Autoinhibition of Dopamine Release May Involve Activation of Potassium (K+) Channels, Pages 265-268, K. Racké, U. Haas, S. Sperb, A. Fischbach, H. Hof, S. Sirrenberg, R. Wammack
3,4-diaminopyridine-evoked Noradrenaline Release in Hippocampal Slices: Further Properties and Involvement of Adenylate Cyclase, Pages 269-270, R. Jackisch, H. Rensing, H.Y. Huang, C. Allgaier, G. Hertting
Interneuronal Cyclic GMP and ‘EDRF-like Substance’ Modulate Norepinephrine Release from Peripheral Sympathetic Nerves, Pages 271-274, S. Greenberg, F.P.J. Diecke, M. Wang, J. Xie, T.P. Tanaka
Modulatory Role of Neuropeptide Y and Peptide YY at the NMDA Receptor Complex, Pages 275-276, F.J. Roman, X. Pascaud, O. Duffy, J.L. Junien
Prejunctional Neuropeptide Y Receptors Are Linked to a G-protein: a Study with N-Ethylmaleimide and Pertussis Toxin, Pages 277-278, S. Foucart, T.V. Murphy, H. Majewski
Protein Kinase C and Modulation of Neurotransmission: Studies With Protein Kinase Inhibitors, Pages 279-280, I.F. Musgrave, H. Majewski
Intrasynaptosomal Protein Phosphorylation and Its Inhibition by Plasma Membrane Oxidoreductases, Pages 281-283, J.-L. Dreyer
Functional and Regulatory Properties of Presynaptic Autoreceptors of the 5-HT1A Subtype on Dorsal Raphe Neurons in Brain Stem Slices, Pages 285-288, L. Lanfumey, S. Haj-Dahmane, L.E. Schechter, F.J. Bolaños, H. Gozlan, M. Hamon
Do Schwann Cells Play a Role in ‘Upstream’ Regulation of the Release Probability in Sympathetic Nerve Varicosities?, Pages 289-292, Lennart Stjärne, Eivor Stjärne, Mussie Msghina, Jian-Xin Bao
Changes in α2 Presynaptic Receptor Sensitivity During Production of Dependence to Morphine in Conscious Rats, Pages 293-296, W.R. Dixon, Juan Machado, Andi P.L. Chang
Role of Presynaptic α2 Heteroreceptors in Nonsynaptic Modulation of Transmitter Release, Pages 297-301, E.S. Vizi, I.J. Elenkov, F. Oberfrank, J. Kiss, L.G. Hársing Jr
Autoregulation of Catecholamine Release at Central and Sympathetic Nerve Terminals: Common Features, Pages 303-306, F. Gonon, M.F. Suaud-Chagny, C. Mermet, L. Stjärne
Autoreceptor Mediated Changes in Dopaminergic Terminal Excitability in vivo, Pages 307-310, J.M. Tepper
Prejunctional Autoreceptors in Mouse vas deferens, Pages 311-314, K. Starke, I. von Kügelgen, R. Bültmann
SK&F 104078 Identifies Subtypes of Prejunctional α2-adrenoceptors in the Rat vas deferens, Pages 315-318, R.R. Ruffolo Jr., A.J. Nichols, J.P. Hieble, M.A. Oriowo
Clonidine Inhibition of Norepinephrine Release from Normal and Morphine-Tolerant Guinea Pig Cortical Slices, Pages 319-322, L. Beani, C. Tomasini, R. Guidorzi, C. Bianchi
Human Caki-1 Cells Are the First Clonal Cell Line Known to Possess the Extraneuronal Transport Mechanism for Noradrenaline (Uptake2), Pages 323-326, E. Schömig, C.-L. Schönfeld, U. Trendelenburg
Inhibition of NA Uptake by (+)-oxaprotiline Inhibits Sympathetic Nerve Activity, Pages 327-328, Andrea Schultheiss, Bela Szabo, Klaus Starke
Autoregulation of Evoked Noradrenaline Release at the Surface of the Isolated Rat Tail Artery Studied by Electrochemistry, Pages 329-330, C. Mermet, L. Stjärne, F. Gonon
Autoregulation of Evoked Noradrenaline Release in the Rat Hypothalamic Paraventricular Nucleus Studied in vivo by Electrochemistry, Pages 331-332, C. Mermet, M.F. Suaud-Chagny, F. Gonon
Clonidine Early in Life: Effect on Brain Morphofunctional Disturbances Induced by Neonatal Malnutrition in the Rat, Pages 333-334, R. Soto-Moyano, A. Hernandez, H. Perez, S. Ruiz, X. Galleguillos, J. Belmar
μ and κ Agonists Inhibit Carbachol-evoked Release of Catecholamines and [Met]enkephalin from ex situ Perfused Dog Adrenals, Pages 335-336, M.K. Dousa, S.L. Chritton, C. Grabau, T.L. Yaksh, G.M. Tyce
Electrophysiological Evidences for the Preferential Location of D2 Autoreceptors on Dendrites of DA Neurons in the Rat Substantia Nigra, Pages 337-338, P.J. Charlety, H. Akaoka, C.F. Saunier, M. Buda, G. Chouvet
Increase of Postsynaptic Dopaminergic Transmission by Presynaptic Actions of Cocaine, Pages 339-340, S.P. Banerjee, C. Manetto, T.I. Lidsky
Autoregulation of Evoked Dopamine Release in the Rat at Central Terminal Sites Studied in vivo by Electrochemistry, Pages 341-342, M.F. Suaud-Chagny, M. Buda, F. Gonon
Combined Effect of (—)-Vesamicol and (+)-Tubocurarine on Endplate Current Amplitude in Rat Skeletal Muscle at High Frequencies of Nerve Stimulation, Pages 343-344, C. Prior, T. Searl, K. Pemberton, W.C. Bowman, I.G. Marshall
Effect of (—)-Vesamicol on Miniature Endplate Current and Endplate Current Amplitudes in Rat Skeletal Muscle, Pages 345-346, T. Searl, C. Prior, I.G. Marshall
Subject Index, Pages 347-352