Drug Design

Content: 
MEDICINAL CHEMISTRY: A Series of Monographs, Page ii
Front Matter, Page iii
Copyright, Page iv
List of Contributors, Pages ix-x
Preface, Page xi, E.J. ARIËNS
Contents of Other Volumes, Pages xiii-xv
Chapter 1 - Microbial Conversion as a Tool in the Preparation of Drugs, Pages 1-131, R. Beukers, A.F. Marx, M.H.J. Zuidweg
Chapter 2 - The Use of Linear Free Energy Parameters and Other Experimental Constants in Structure–Activity Studies, Pages 133-187, A. Verloop
Chapter 3 - Anticoagulants Structurally and Functionally Related to Vitamin K, Pages 189-203, T. Kralt, V. Claassen
Chapter 4 - Design of β-Blocking Drugs, Pages 205-228, A.M. Barrett
Chapter 5 - The Design of Biologically Active Acridines, Pages 229-242, Adrien Albert
Chapter 6 - The Design of Local Anesthetics, Pages 243-391, J. Büchi, X. Perlia
Chapter 7 - Design of Insect Chemosterilants, Pages 393-413, Ralph B. Turner
Chapter 8 - Molecular Approach for Designing Inhibitors to Enzymes Involved in Blood Clotting, Pages 415-447, L. Lorandand, J.L.G. Nilsson
Author Index, Pages 449-473
Subject Index, Pages 475-502